BDBM50192163 (R,E)-N-(1-cinnamylpyrrolidin-3-yl)-3,5-dimethoxybenzamide::CHEMBL215114

SMILES COc1cc(OC)cc(c1)C(=O)N[C@@H]1CCN(C\C=C\c2ccccc2)C1

InChI Key InChIKey=KUNCBFJZBIUEAD-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50192163   

TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192163((R,E)-N-(1-cinnamylpyrrolidin-3-yl)-3,5-dimethoxyb...)
Affinity DataKi:  17nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192163((R,E)-N-(1-cinnamylpyrrolidin-3-yl)-3,5-dimethoxyb...)
Affinity DataIC50: 42nMAssay Description:Inhibition of MCH-mediated calcium release by CHO cells expressing human MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed