BDBM50193879 CHEMBL218656::N-(4-(2-(diethylamino)ethoxy)phenyl)-7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-amine::US8481536, 364

SMILES CCN(CC)CCOc1ccc(Nc2nnc3cc(cc(C)c3n2)-c2c(C)cccc2C)cc1

InChI Key InChIKey=BWIWBRIZCJKRBV-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50193879   

TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

US Patent
LigandPNGBDBM50193879(US8481536, 364 | CHEMBL218656 | N-(4-(2-(diethylam...)
Affinity DataIC50: 9.67nMT: 2°CAssay Description:Recombinant human c-Src or Yes (28 ng/well, Panvera/Invitrogen, Madison Wis.), ATP (3 μM), a tyrosine kinase substrate (PTK2, 250 μM, Promega C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2013
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

US Patent
LigandPNGBDBM50193879(US8481536, 364 | CHEMBL218656 | N-(4-(2-(diethylam...)
Affinity DataIC50: 10nMAssay Description:Inhibition of SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

US Patent
LigandPNGBDBM50193879(US8481536, 364 | CHEMBL218656 | N-(4-(2-(diethylam...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed