BDBM50197710 CHEMBL3959997

SMILES Cc1cc2cc(-n3ncc(C(=O)c4cc5ccccc5[nH]4)c3N)ccc2[nH]1

InChI Key InChIKey=QIASHDRGDBMNGW-UHFFFAOYSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50197710   

TargetVascular endothelial growth factor receptor 2(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197710BDBM50197710(CHEMBL3959997)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of human KDR by time-resolved fluorescence or time-resolved fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2018
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 3(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197710BDBM50197710(CHEMBL3959997)
Affinity DataIC50: 18nMAssay Description:Inhibition of human FGFR3 by time-resolved fluorescence or time-resolved fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2018
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197710BDBM50197710(CHEMBL3959997)
Affinity DataIC50: 32nMAssay Description:Inhibition of human FGFR2 by time-resolved fluorescence or time-resolved fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2018
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 1(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197710BDBM50197710(CHEMBL3959997)
Affinity DataIC50: 69nMAssay Description:Inhibition of human FGFR1 by time-resolved fluorescence or time-resolved fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2018
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 4(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197710BDBM50197710(CHEMBL3959997)
Affinity DataIC50: 85nMAssay Description:Inhibition of human FGFR4 by time-resolved fluorescence or time-resolved fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2018
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197710BDBM50197710(CHEMBL3959997)
Affinity DataIC50: 330nMAssay Description:Inhibition of human SRC by time-resolved fluorescence or time-resolved fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2018
Entry Details Article
PubMed