BDBM50202686 7-fluoro-4-oxo-N-(1-((3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)methyl)piperidin-4-yl)-4H-chromene-2-carboxamide::CHEMBL217233

SMILES Fc1ccc2c(c1)oc(cc2=O)C(=O)NC1CCN(Cc2ccc3OCC(=O)Nc3c2)CC1

InChI Key InChIKey=GOGGRAWNDKPWNO-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50202686   

TargetMelanin-concentrating hormone receptor 1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50202686(7-fluoro-4-oxo-N-(1-((3-oxo-3,4-dihydro-2H-benzo[b...)
Affinity DataIC50: 19nMAssay Description:Displacement of 125I-MCH from MCH-R1 expressed in IMR-32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50202686(7-fluoro-4-oxo-N-(1-((3-oxo-3,4-dihydro-2H-benzo[b...)
Affinity DataIC50: 5.79E+3nMAssay Description:Displacement of 3H-dofetilide from hERG-expressing HEK membrane homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed