BDBM50224214 2-(1H-indazol-5-ylamino)-5-isopropylthiazol-4(5H)-one::CHEMBL238975

SMILES CC(C)c1sc(Nc2ccc3n[nH]cc3c2)nc1O

InChI Key InChIKey=AZCHUDGHZUVLTF-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50224214   

LigandPNGBDBM50224214(2-(1H-indazol-5-ylamino)-5-isopropylthiazol-4(5H)-...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50224214(2-(1H-indazol-5-ylamino)-5-isopropylthiazol-4(5H)-...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human 11-beta-HSD1 in CHO cells assessed as conversion of cortisone to cortisolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed