BDBM50224408 8-bromo-3-(4-chloro-phenyl)-9-methylamino-3H-pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-one::CHEMBL241547

SMILES CNc1c(Br)cnc2sc3c(ncn(-c4ccc(Cl)cc4)c3=O)c12

InChI Key InChIKey=PFKFGKXVMKQDJI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50224408   

TargetMetabotropic glutamate receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50224408(8-bromo-3-(4-chloro-phenyl)-9-methylamino-3H-pyrid...)
Affinity DataIC50: 5.90nMAssay Description:Antagonist activity at human mGluR1a expressed in CHO cells assessed by measuring intracellular calcium by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed