BDBM50228648 5,7-dichloro-3-(3-hydroxyphenyl)-3-methylquinoline-2,4(1H,3H)-dione::CHEMBL404352

SMILES CC1(C(=O)Nc2cc(Cl)cc(Cl)c2C1=O)c1cccc(O)c1

InChI Key InChIKey=MUALJDCOWOWPTA-UHFFFAOYSA-N

Data  9 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 50228648   

Target5-hydroxytryptamine receptor 6(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50228648(5,7-dichloro-3-(3-hydroxyphenyl)-3-methylquinoline...)
Affinity DataKi:  30.1nMAssay Description:Displacement of [3H]LSD from human cloned 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50228648(5,7-dichloro-3-(3-hydroxyphenyl)-3-methylquinoline...)
Affinity DataKi:  1.81E+3nMAssay Description:Displacement of [3H]SCH-23390 from human cloned dopamine D1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50228648(5,7-dichloro-3-(3-hydroxyphenyl)-3-methylquinoline...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50228648(5,7-dichloro-3-(3-hydroxyphenyl)-3-methylquinoline...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50228648(5,7-dichloro-3-(3-hydroxyphenyl)-3-methylquinoline...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50228648(5,7-dichloro-3-(3-hydroxyphenyl)-3-methylquinoline...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50228648(5,7-dichloro-3-(3-hydroxyphenyl)-3-methylquinoline...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50228648(5,7-dichloro-3-(3-hydroxyphenyl)-3-methylquinoline...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50228648(5,7-dichloro-3-(3-hydroxyphenyl)-3-methylquinoline...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed