BDBM50231108 CHEMBL253014::N-(2-chlorophenethyl)-4-(trifluoromethoxy)benzamide

SMILES FC(F)(F)Oc1ccc(cc1)C(=O)NCCc1ccccc1Cl

InChI Key InChIKey=VEMICVMDQMTCNQ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50231108   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50231108(N-(2-chlorophenethyl)-4-(trifluoromethoxy)benzamid...)Copy SMILESCopy InChI

Affinity DataIC50: 776nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced calcium influx in HEK293 cellsMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
Entry Details Article
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