BDBM50232124 1-(5-tert-butyl-2,2-difluoro-2,3-dihydro-1H-inden-1-yl)-3-(1H-indazol-4-yl)urea::CHEMBL254019

SMILES CC(C)(C)c1ccc2C(NC(=O)Nc3cccc4[nH]ncc34)C(F)(F)Cc2c1

InChI Key InChIKey=BGZQKFANVOPJDS-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50232124   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50232124(1-(5-tert-butyl-2,2-difluoro-2,3-dihydro-1H-inden-...)Copy SMILESCopy InChI

Affinity DataIC50: 216nMAssay Description:Blockade of human TRPV1 receptor assessed as inhibition of capsaicin-induced calcium fluxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
Entry Details Article
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