BDBM50232567 CHEMBL4067234

SMILES Fc1ccc2sc(COc3cccc(c3)C(=O)NCc3ccc(cc3)C(=O)NS(=O)(=O)c3cccc(Cl)c3)nc2c1

InChI Key InChIKey=DHEDSOOHLBLFHH-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50232567   

TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Askat

Curated by ChEMBL
LigandPNGBDBM50232567(CHEMBL4067234)
Affinity DataIC50:  302nMAssay Description:Antagonist activity at human EP4 receptor expressed in HEK293 cells assessed as inhibition of PGE2-induced cAMP level by HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed