BDBM50234102 CHEMBL4090052

SMILES OC(=O)[C@@H]1C[C@H](CN1)Oc1cc2ccccc2cc1C(O)=O

InChI Key InChIKey=DHPQJRYFIYLEEK-UHFFFAOYSA-N

Data  5 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50234102   

TargetGlutamate receptor ionotropic, kainate 1(Rat)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234102(CHEMBL4090052)
Affinity DataKi:  3.50E+3nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2019
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 1(Rat)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234102(CHEMBL4090052)
Affinity DataKi:  3.51E+3nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2019
Entry Details Article
PubMed
TargetGlutamate receptor 2(Rat)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234102(CHEMBL4090052)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of (RS)-[3H]AMPA from eGFP-fused recombinant rat full length GluA2 receptor expressed in HEK293T/17 cells by liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2019
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234102(CHEMBL4090052)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK3 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2019
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234102(CHEMBL4090052)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK2 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2019
Entry Details Article
PubMed