BDBM50234110 CHEMBL4090961

SMILES CC(=O)c1ccc(O[C@H]2CN[C@@H](C2)C(O)=O)c(c1)C(O)=O

InChI Key InChIKey=KAZFDFAPKWRBAV-UHFFFAOYSA-N

Data  6 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50234110   

TargetGlutamate receptor ionotropic, kainate 1(Rat)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234110(CHEMBL4090961)
Affinity DataKi:  4.68E+3nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2019
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 1(Rat)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234110(CHEMBL4090961)
Affinity DataKi:  4.70E+3nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2019
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234110(CHEMBL4090961)
Affinity DataKi:  2.95E+4nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK3 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2019
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234110(CHEMBL4090961)
Affinity DataKi:  3.00E+4nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK3 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2019
Entry Details Article
PubMed
TargetGlutamate receptor 2(Rat)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234110(CHEMBL4090961)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of (RS)-[3H]AMPA from eGFP-fused recombinant rat full length GluA2 receptor expressed in HEK293T/17 cells by liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2019
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234110(CHEMBL4090961)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK2 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2019
Entry Details Article
PubMed