BDBM50238820 CHEMBL4072676

SMILES CNc1ncc2cc(-c3cc(OC)cc(OC)c3Cl)c(=O)n(CCc3ccc(cc3)N(C)C(=O)C=C)c2n1

InChI Key InChIKey=WGLICLJLEWRTIS-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50238820   

TargetFibroblast growth factor receptor 1(Human)
Principia Biopharma

Curated by ChEMBL
LigandPNGBDBM50238820(CHEMBL4072676)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human FGFR1 using 5-FAM-KKKKEEIYFFF-NH2 as substrate preincubated for 15 mins followed by peptide substrate addition measured after 3 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2019
Entry Details Article
PubMed