BDBM50238933 CHEMBL4089962

SMILES CC(C)(C)c1ccc(Oc2cccc(COc3ccccc3CCC(=O)OCCCOP(O)(=O)OC[C@H](N)C(O)=O)c2)cc1

InChI Key InChIKey=HGYBEZUXJPBXOR-NDEPHWFRSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50238933   

TargetProbable G-protein coupled receptor 34(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50238933(CHEMBL4089962)
Affinity DataEC50:  900nMAssay Description:Opioid receptor mu 1 affinity against the receptor site model site 1 (mu1) by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 34(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50238933(CHEMBL4089962)
Affinity DataEC50:  295nMAssay Description:Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of AP-TGFalpha re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 34(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50238933(CHEMBL4089962)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of AP-TGFalpha re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 34(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50238933(CHEMBL4089962)
Affinity DataEC50:  912nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of ectodomain she...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed