BDBM50238989 CHEMBL4087337

SMILES COc1ccc2O\C(=C/c3ccc(O)c(O)c3)C(=O)c2c1

InChI Key InChIKey=IOJLBZJSULGZLY-UHFFFAOYSA-N

Data  11 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 11 hits for monomerid = 50238989   

TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 510nMAssay Description:Inhibition of human TEKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetAurora kinase A(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of human AURORA-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 2.19E+3nMAssay Description:Inhibition of human ITKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase Blk(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 3.05E+3nMAssay Description:Inhibition of human BLKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 5.03E+3nMAssay Description:Inhibition of human BTKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17A(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 5.81E+3nMAssay Description:Inhibition of human DRAK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDeath-associated protein kinase 2(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 6.34E+3nMAssay Description:Inhibition of human DAPK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 8.84E+3nMAssay Description:Inhibition of human CDK5More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDeath-associated protein kinase 3(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of human DAPK3More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed