BDBM50249083 CHEMBL473992::N-Adamantan-1-yl-3-{[2-(4-bromo-3-methyl-phenoxy)-acetyl]-hydrazono}-butyramide

SMILES CC(CC(=O)NC12CC3CC(CC(C3)C1)C2)=NNC(=O)COc1ccc(Br)c(C)c1

InChI Key

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50249083   

Target11-beta-hydroxysteroid dehydrogenase 1(Mouse)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50249083(N-Adamantan-1-yl-3-{[2-(4-bromo-3-methyl-phenoxy)-...)
Affinity DataIC50: 6.55E+3nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in HEK293 cells assessed as conversion of [3H]cortisone to [3H]cortisol by scintillation proximity assay in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50249083(N-Adamantan-1-yl-3-{[2-(4-bromo-3-methyl-phenoxy)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells assessed as conversion of [3H]cortisone to [3H]cortisol by scintillation proximity assay in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed