BDBM50251648 CHEMBL479952::N-(6-(pyridin-3-yloxy)pyridin-3-yl)-1H-indole-3-carboxamide

SMILES O=C(Nc1ccc(Oc2cccnc2)nc1)c1c[nH]c2ccccc12

InChI Key InChIKey=BVEOZKOLIKNPKQ-UHFFFAOYSA-N

Data  8 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50251648   

Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50251648(N-(6-(pyridin-3-yloxy)pyridin-3-yl)-1H-indole-3-ca...)
Affinity DataIC50: 1.60nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50251648(N-(6-(pyridin-3-yloxy)pyridin-3-yl)-1H-indole-3-ca...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50251648(N-(6-(pyridin-3-yloxy)pyridin-3-yl)-1H-indole-3-ca...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]LSD from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50251648(N-(6-(pyridin-3-yloxy)pyridin-3-yl)-1H-indole-3-ca...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50251648(N-(6-(pyridin-3-yloxy)pyridin-3-yl)-1H-indole-3-ca...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50251648(N-(6-(pyridin-3-yloxy)pyridin-3-yl)-1H-indole-3-ca...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50251648(N-(6-(pyridin-3-yloxy)pyridin-3-yl)-1H-indole-3-ca...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]LSD from human cloned 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50251648(N-(6-(pyridin-3-yloxy)pyridin-3-yl)-1H-indole-3-ca...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed