BDBM50256810 CHEMBL508680::trans-[2-(6-Chloro-2-fluoro-3-methylphenyl)cyclopropyl]methylamineHydrochloride

SMILES Cc1ccc(Cl)c([C@H]2C[C@@H]2CN)c1F

InChI Key InChIKey=KKDCPAICZNOUFD-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50256810   

Target5-hydroxytryptamine receptor 2C(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50256810(trans-[2-(6-Chloro-2-fluoro-3-methylphenyl)cyclopr...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50256810(trans-[2-(6-Chloro-2-fluoro-3-methylphenyl)cyclopr...)
Affinity DataEC50:  116nMAssay Description:Agonist activity at human 5HT2B receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50256810(trans-[2-(6-Chloro-2-fluoro-3-methylphenyl)cyclopr...)
Affinity DataEC50:  330nMAssay Description:Agonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed