BDBM50257781 2-(3-(3-methoxyphenyl)-3-methylazetidin-1-yl)pyridin-4-amine::CHEMBL492909

SMILES COc1cccc(c1)C1(C)CN(C1)c1cc(N)ccn1

InChI Key InChIKey=PSAGNQSIEQQFKW-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50257781   

TargetDelta-type opioid receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50257781(2-(3-(3-methoxyphenyl)-3-methylazetidin-1-yl)pyrid...)
Affinity DataEC50:  846nMAssay Description:Agonist activity at delta opioid receptor expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP production by ALPHAscreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50257781(2-(3-(3-methoxyphenyl)-3-methylazetidin-1-yl)pyrid...)
Affinity DataKi:  1.84E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed