BDBM50257889 1-(1-(4-aminopyridin-2-yl)-4-phenylpiperidin-4-yl)ethanone::CHEMBL494771

SMILES CC(=O)C1(CCN(CC1)c1cc(N)ccn1)c1ccccc1

InChI Key InChIKey=HHUZCRCCGCQHQE-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50257889   

TargetDelta-type opioid receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50257889(1-(1-(4-aminopyridin-2-yl)-4-phenylpiperidin-4-yl)...)
Affinity DataEC50:  263nMAssay Description:Agonist activity at delta opioid receptor expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP production by ALPHAscreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50257889(1-(1-(4-aminopyridin-2-yl)-4-phenylpiperidin-4-yl)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed