BDBM50258161 2-(4-tert-butylphenyl)-4-(4-((1,3,5-trimethyl-1H-pyrazol-4-yl)methyl)piperazin-1-yl)-1H-benzo[d]imidazole::CHEMBL495190

SMILES Cc1nn(C)c(C)c1CN1CCN(CC1)c1cccc2[nH]c(nc12)-c1ccc(cc1)C(C)(C)C

InChI Key InChIKey=CMKDKQAMZWVGKC-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50258161   

TargetGonadotropin-releasing hormone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50258161(2-(4-tert-butylphenyl)-4-(4-((1,3,5-trimethyl-1H-p...)
Affinity DataIC50: 38nMAssay Description:Displacement of [125I]-(D-Trp6)-GnRH from human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50258161(2-(4-tert-butylphenyl)-4-(4-((1,3,5-trimethyl-1H-p...)
Affinity DataIC50: 450nMAssay Description:Displacement of [125I]-(D-Trp6)-GnRH from rat GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed