BDBM50261384 CHEMBL526550::H-DPhe2-c[Ncy3-Phe7-DTrp8-Lys9-Thr10-Ncy14]-Thr15-NH2

SMILES C[C@@H](O)[C@H](NC(=O)[C@@H]1NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](NC(=O)[C@H](N)Cc2ccccc2)SS1)[C@@H](C)O)C(N)=O

InChI Key InChIKey=OWUWTNRTKGNXIY-UHFFFAOYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50261384   

TargetSomatostatin receptor type 4(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50261384(H-DPhe2-c[Ncy3-Phe7-DTrp8-Lys9-Thr10-Ncy14]-Thr15-...)
Affinity DataIC50: 214nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]SRIF28 from human sst4 receptor expressed in chinese hamster CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50261384(H-DPhe2-c[Ncy3-Phe7-DTrp8-Lys9-Thr10-Ncy14]-Thr15-...)
Affinity DataIC50: 337nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]SRIF28 from human sst2 receptor expressed in chinese hamster CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50261384(H-DPhe2-c[Ncy3-Phe7-DTrp8-Lys9-Thr10-Ncy14]-Thr15-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]SRIF28 from human sst3 receptor expressed in chinese hamster CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50261384(H-DPhe2-c[Ncy3-Phe7-DTrp8-Lys9-Thr10-Ncy14]-Thr15-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]SRIF28 from human sst1 receptor expressed in CHOK1 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50261384(H-DPhe2-c[Ncy3-Phe7-DTrp8-Lys9-Thr10-Ncy14]-Thr15-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]SRIF28 from human sst5 receptor expressed in CHOK1 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed