BDBM50262132 CHEMBL468409::methyl 2-(4-bromophenyl)-5-((3-(5,6-dimethyl-1H-benzo[d]imidazol-2-yl)propyl)(methyl)amino)-2-isopropylpentanoate

SMILES COC(=O)C(CCCN(C)CCCc1nc2cc(C)c(C)cc2[nH]1)(C(C)C)c1ccc(Br)cc1

InChI Key InChIKey=PPUATJSILURJNL-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50262132   

TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50262132(methyl 2-(4-bromophenyl)-5-((3-(5,6-dimethyl-1H-be...)
Affinity DataIC50: 53.0nMAssay Description:Antagonist activity at T type calcium channel alpha1G expressed in HEK293 cells assessed as inhibition of peak currents by whole-cell patch-clamp met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed