BDBM50264702 CHEMBL489400::N-(4-Chlorophenyl)-1-(3-(trifluoromethyl)pyridin-2-yl)-1,2,3,6-tetrahydropyridine-4-carboxamide

SMILES FC(F)(F)c1cccnc1N1CCC(=CC1)C(=O)Nc1ccc(Cl)cc1

InChI Key InChIKey=BHBZFJBSLMYUOQ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50264702   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50264702(N-(4-Chlorophenyl)-1-(3-(trifluoromethyl)pyridin-2...)Copy SMILESCopy InChI

Affinity DataIC50: 19nMAssay Description:Antagonist activity at human recombinant TRPV1 expressed in human 1321N1 cells assessed as inhibition of capsaicin-induced calcium influx by FLIPR as...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
1/11/2010
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL