BDBM50265881 CHEMBL4065890

SMILES OC(=O)CCc1ccc(cc1)-c1ccc2c(nn(-c3ccccn3)c2c1)C#N

InChI Key InChIKey=WTZBWVUYQRHSRU-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50265881   

TargetFree fatty acid receptor 1(Mouse)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265881(CHEMBL4065890)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at mouse GPR40 expressed in HEK293 cells assessed as increase in intracellular calcium level after 5 mins by FLUO-4-AM dye-based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265881(CHEMBL4065890)
Affinity DataEC50:  4.80E+3nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed