BDBM50269137 CHEMBL4099561

SMILES O=C(Nc1ccccc1N1CCOCC1)\C=C\c1cccc2cccnc12

InChI Key InChIKey=MYVUHXRZRNJGSU-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50269137   

TargetSodium channel protein type 9 subunit alpha(Human)
Amgen

Curated by ChEMBL

LigandBDBM50269137(CHEMBL4099561)Copy SMILESCopy InChI

Affinity DataIC50: 43nMAssay Description:Inhibition of slow inactivated human NaV1.7 expressed in HEK293 cells at -20 mV holding potential after 5 mins by IonWorks electrophysiology methodMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
3/9/2020
Entry Details Article
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