BDBM50273253 3-(7-(3-(trifluoromethyl)pyridin-2-yl)-4-(6-(trifluoromethyl)pyridin-3-ylamino)quinazolin-2-yl)propanoic acid::CHEMBL515050

SMILES OC(=O)CCc1nc(Nc2ccc(nc2)C(F)(F)F)c2ccc(cc2n1)-c1ncccc1C(F)(F)F

InChI Key InChIKey=XUJHWPHTWPTVGT-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50273253   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen

Curated by ChEMBL

LigandBDBM50273253(3-(7-(3-(trifluoromethyl)pyridin-2-yl)-4-(6-(trifl...)Copy SMILESCopy InChI

Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at human TRPV1 receptor assessed as inhibition of capsaicin-induced activationMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
1/11/2010
Entry Details Article
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