BDBM50276182 CHEMBL4128521

SMILES COC[C@@H]1CCCN1Cc1cc(ccc1-c1ccccc1)C(=O)Nc1ccc2CCC(=O)N(C)c2c1

InChI Key InChIKey=KETNHMSQZQWLHN-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50276182   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Astellas Pharma

Curated by ChEMBL

LigandBDBM50276182(CHEMBL4128521)Copy SMILESCopy InChI

Affinity DataIC50: 150nMAssay Description:Displacement of [3H]RTX from human TRPV1 expressed in HEK293 cell membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
5/22/2020
Entry Details Article
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