BDBM50278254 5-(4-bromophenyl)-3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-1-(2,4-dichlorophenyl)-N-phenyl-1H-pyrazole-4-carboxamide::CHEMBL469771

SMILES CC(C)(C)c1nnc(o1)-c1nn(c(c1C(=O)Nc1ccccc1)-c1ccc(Br)cc1)-c1ccc(Cl)cc1Cl

InChI Key InChIKey=UVFWCIGTUOMCPO-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50278254   

TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278254(5-(4-bromophenyl)-3-(5-tert-butyl-1,3,4-oxadiazol-...)
Affinity DataIC50: 1.35nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278254(5-(4-bromophenyl)-3-(5-tert-butyl-1,3,4-oxadiazol-...)
Affinity DataIC50: 386nMAssay Description:Displacement of [3H]WIN-55212-2 from human recombinant cannabinoid CB2 receptor expressed in CHOK1 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed