BDBM50278708 CHEMBL4173280

SMILES OC(=O)CCc1cc(F)c(OCc2c(nsc2C(F)(F)F)-c2ccc(cc2)C#N)c(F)c1

InChI Key InChIKey=HNYQVJLQRVUHLH-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50278708   

TargetFree fatty acid receptor 4(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50278708(CHEMBL4173280)
Affinity DataEC50:  332nMAssay Description:Agonist activity at PK-tagged human GPR120 long isoform expressed in CHOK1 cells co-expressing EA-tagged beta-arrestin assessed as beta-gal enzyme co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50278708(CHEMBL4173280)
Affinity DataEC50:  672nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux incubated for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2020
Entry Details Article
PubMed