BDBM50297594 1-(cyclopropylmethyl)-5-(2-methoxyethylsulfonyl)-2-neopentyl-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridine::CHEMBL560208

SMILES COCCS(=O)(=O)N1CCc2c(C1)nc(CC(C)(C)C)n2CC1CC1

InChI Key InChIKey=WHFDUZQMHSPVLQ-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50297594   

TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50297594(1-(cyclopropylmethyl)-5-(2-methoxyethylsulfonyl)-2...)
Affinity DataEC50:  21.5nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50297594(1-(cyclopropylmethyl)-5-(2-methoxyethylsulfonyl)-2...)
Affinity DataEC50:  1.40E+4nMAssay Description:Agonist activity at human recombinant CB1 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed