BDBM50300424 CHEMBL572965::Methyl 3-(5-chloro-4-methyl-3-oxoisothiazol-2(3H)-yl)propanoate

SMILES COC(=O)CCn1sc(Cl)c(C)c1=O

InChI Key InChIKey=YETKKDGVXTZNOU-UHFFFAOYSA-N

Data  1 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50300424   

TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50300424(Methyl 3-(5-chloro-4-methyl-3-oxoisothiazol-2(3H)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant histone acetyltransferase PCAF assessed as CoA-SH activity preincubated for 15 mins by CPM fluorescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed