BDBM50305421 1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanomethyl)-N-morpholino-1H-pyrazole-3-carboxamide::CHEMBL604061

SMILES Clc1ccc(cc1)-c1c(CC#N)c(nn1-c1ccccc1Cl)C(=O)NN1CCOCC1

InChI Key InChIKey=SPUWBWJYUKCTKB-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50305421   

TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305421(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 71nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-induced GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305421(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 71nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed