BDBM50305986 5,6-bis(4-chlorophenyl)-N-cyclohexylpyrazine-2-carbothioamide::CHEMBL611057

SMILES Clc1ccc(cc1)-c1ncc(nc1-c1ccc(Cl)cc1)C(=S)NC1CCCCC1

InChI Key InChIKey=HLJFBDANUXYSFO-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50305986   

TargetCannabinoid receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50305986(5,6-bis(4-chlorophenyl)-N-cyclohexylpyrazine-2-car...)
Affinity DataIC50: 5.80nMAssay Description:Agonist activity at human CB1 receptor assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed