BDBM50308577 1-(4-Fluorophenyl)-8-{[(2-morpholin-4-ylpyridin-3-yl)carbonyl]amino}-4,5-dihydro-1H-benzo[g]indazole-3-carboxamide::CHEMBL589808

SMILES NC(=O)c1nn(c-2c1CCc1ccc(NC(=O)c3cccnc3N3CCOCC3)cc-21)-c1ccc(F)cc1

InChI Key InChIKey=IGRCHSUORINQGN-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50308577   

TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50308577(1-(4-Fluorophenyl)-8-{[(2-morpholin-4-ylpyridin-3-...)Copy SMILESCopy InChI

Affinity DataIC50: 1.42E+4nMAssay Description:Inhibition of human recombinant IKK2-mediated transfer of [gamma33P]ATP to biotinylated IkappaBalpha after 30 mins by scintillation countingMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
9/2/2010
Entry Details Article
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