BDBM50321461 2-bromo-N-(2,5-dichlorothiophen-3-ylsulfonyl)-N-phenylacetamide::CHEMBL1171238

SMILES Clc1cc(c(Cl)s1)S(=O)(=O)N(C(=O)CBr)c1ccccc1

InChI Key InChIKey=XOLGJVQMYMQCNT-UHFFFAOYSA-N

Data  9 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 50321461   

TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research

Curated by ChEMBL
LigandPNGBDBM50321461(2-bromo-N-(2,5-dichlorothiophen-3-ylsulfonyl)-N-ph...)
Affinity DataIC50: 600nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Montclair State University

Curated by ChEMBL
LigandPNGBDBM50321461(2-bromo-N-(2,5-dichlorothiophen-3-ylsulfonyl)-N-ph...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human CDK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Montclair State University

Curated by ChEMBL
LigandPNGBDBM50321461(2-bromo-N-(2,5-dichlorothiophen-3-ylsulfonyl)-N-ph...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human CDK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
Montclair State University

Curated by ChEMBL
LigandPNGBDBM50321461(2-bromo-N-(2,5-dichlorothiophen-3-ylsulfonyl)-N-ph...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human CDK6More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 7(Human)
Montclair State University

Curated by ChEMBL
LigandPNGBDBM50321461(2-bromo-N-(2,5-dichlorothiophen-3-ylsulfonyl)-N-ph...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human CDK7More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Walter Reed Army Institute of Research

Curated by ChEMBL
LigandPNGBDBM50321461(2-bromo-N-(2,5-dichlorothiophen-3-ylsulfonyl)-N-ph...)
Affinity DataIC50: 2.15E+4nMAssay Description:Inhibition of human CDK1/cyclin BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
Walter Reed Army Institute of Research

Curated by ChEMBL
LigandPNGBDBM50321461(2-bromo-N-(2,5-dichlorothiophen-3-ylsulfonyl)-N-ph...)
Affinity DataIC50: 2.85E+4nMAssay Description:Inhibition of human CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Human)
Walter Reed Army Institute of Research

Curated by ChEMBL
LigandPNGBDBM50321461(2-bromo-N-(2,5-dichlorothiophen-3-ylsulfonyl)-N-ph...)
Affinity DataIC50: 3.34E+4nMAssay Description:Inhibition of human CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Walter Reed Army Institute of Research

Curated by ChEMBL
LigandPNGBDBM50321461(2-bromo-N-(2,5-dichlorothiophen-3-ylsulfonyl)-N-ph...)
Affinity DataIC50: 3.49E+4nMAssay Description:Inhibition of human CDK6/Cyclin D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed