BDBM50337990 1-(6-tert-butyl-1-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-3-(1H-indazol-4-yl)urea::CHEMBL1684248

SMILES CN1CCC(NC(=O)Nc2cccc3[nH]ncc23)c2cc(ccc12)C(C)(C)C

InChI Key InChIKey=BGKQAJKETVAKOI-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50337990   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50337990(1-(6-tert-butyl-1-methyl-1,2,3,4-tetrahydroquinoli...)Copy SMILESCopy InChI

Affinity DataIC50: 853nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of calcium influxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
8/24/2011
Entry Details Article
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