BDBM50337998 (R)-1-(1H-indazol-4-yl)-3-(7-(trifluoromethyl)chroman-4-yl)urea::CHEMBL1684271

SMILES FC(F)(F)c1ccc2[C@@H](CCOc2c1)NC(=O)Nc1cccc2[nH]ncc12

InChI Key InChIKey=LNRLQTQYVBBJBO-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50337998   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50337998((R)-1-(1H-indazol-4-yl)-3-(7-(trifluoromethyl)chro...)Copy SMILESCopy InChI

Affinity DataIC50: 4nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of calcium influxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
8/24/2011
Entry Details Article
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