BDBM50340101 CHEMBL1762819::N-(2-fluoroethyl)-8-(6-methoxy-2-methylpyridin-3-yl)-N-(2-methoxyethyl)-2,7-dimethylpyrazolo[1,5-a][1,3,5]triazin-4-amine

SMILES COCCN(CCF)c1nc(C)nc2c(c(C)nn12)-c1ccc(OC)nc1C

InChI Key InChIKey=VGPMUJRKFXDSJW-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50340101   

TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50340101(N-(2-fluoroethyl)-8-(6-methoxy-2-methylpyridin-3-y...)
Affinity DataIC50: 5.5nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed