BDBM50344369 CHEMBL1779833::N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(7-hydroxynaphthalen-1-yl)acetamide

SMILES Oc1ccc2cccc(CC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c2c1

InChI Key InChIKey=STNILISHSOEFAG-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50344369   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Bayer Yakuhin

Curated by ChEMBL

LigandBDBM50344369(N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(7-hydrox...)Copy SMILESCopy InChI

Affinity DataIC50: 34nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
12/4/2011
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL