BDBM50347759 CHEMBL1803070

SMILES CN1C(=O)C(=Cc2ccc3c(c2)OCO3)N=C1Nc1ccc(O)cc1

InChI Key InChIKey=MMWGSUYGZVUNCC-UHFFFAOYSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50347759   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Universite£? De Rennes 1

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347759BDBM50347759(CHEMBL1803070)
Affinity DataIC50: 440nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using KKISGRLSPIMTEQ as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
Universite£? De Rennes 1

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347759BDBM50347759(CHEMBL1803070)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mouse recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Human)
Universite£? De Rennes 1

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347759BDBM50347759(CHEMBL1803070)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human recombinant GST-tagged DYRK2 using KKISGRLSPIMTEQ as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Universite£? De Rennes 1

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347759BDBM50347759(CHEMBL1803070)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK3(Mouse)
Universite£? De Rennes 1

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347759BDBM50347759(CHEMBL1803070)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of mouse recombinant GST-tagged CLK3 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Universite£? De Rennes 1

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347759BDBM50347759(CHEMBL1803070)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human recombinant Pim1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed