BDBM50354641 CHEMBL1834203

SMILES COc1ccc(NC(=O)Nc2ccc(nc2)-c2ccc(cc2)C(=O)N[C@@H](C(C)C)C(O)=O)cc1

InChI Key InChIKey=OWFDKHQRFPSFTJ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50354641   

TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50354641(CHEMBL1834203)
Affinity DataIC50: 25nMAssay Description:Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed