BDBM50362788 CHEMBL1940214

SMILES C[C@H](C(=O)NCCCc1ccc(C)c(C)c1)c1ccc(NS(C)(=O)=O)c(F)c1

InChI Key InChIKey=JYJFYPANGZFUDB-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50362788   

TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362788(CHEMBL1940214)
Affinity DataKi:  33.7nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362788(CHEMBL1940214)
Affinity DataKi:  97nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362788(CHEMBL1940214)
Affinity DataKi:  257nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362788(CHEMBL1940214)
Affinity DataKi:  413nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed