BDBM50376270 CHEMBL406573

SMILES O=C(Nc1cnc2ccccc2c1)c1ccc(NC2CCCCC2)cc1

InChI Key InChIKey=SWEAAERORIFOIX-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50376270   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50376270(CHEMBL406573)
Affinity DataKi:  156nMAssay Description:Displacement of [3H]RTX from human TRPV1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50376270(CHEMBL406573)
Affinity DataIC50: 1.00E+4nMAssay Description:Activity at human TRPV1 in HEK cells assessed by measuring capsaicin-induced calcium level by FLIPR technologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed