BDBM50379275 CHEMBL2011500
SMILES COc1ccc(cc1)C(=O)CC1(O)C(=O)Nc2c1c(Cl)ccc2Cl
InChI Key InChIKey=HLXSCTYHLQHQDJ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50379275
Affinity DataKd: 9.48E+3nMAssay Description:Inhibition of interaction of EWS-Fli1 to GST-tagged RNA Helicase A (647-1075) by surface plasmon resonanceMore data for this Ligand-Target Pair
TargetFriend leukemia integration 1 transcription factor(Human)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of transcriptional activity of full-length EWS-FLI1 (unknown origin) expressed in COS7 cells by NR0B1-luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.74E+4nMAssay Description:Binding affinity to ETV1 by surface plasmon resonanceMore data for this Ligand-Target Pair
Affinity DataKd: 1.17E+4nMAssay Description:Binding affinity to ERG by surface plasmon resonanceMore data for this Ligand-Target Pair