BDBM50387017 CHEMBL2049193

SMILES CCCN(CCC)c1cccc2nc(Nc3c(C)cc(C)cc3C)c(C)cc12

InChI Key InChIKey=RBYNVYWHUQMOGA-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50387017   

LigandPNGBDBM50387017(CHEMBL2049193)
Affinity DataIC50: 88nMAssay Description:Displacement of [125I]-CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandPNGBDBM50387017(CHEMBL2049193)
Affinity DataIC50: 372nMAssay Description:Antagonist activity at human CRF1 receptor expressed in HEK293 cells assessed as inhibition of CRF-stimulated intracellular cAMP accumulation preincu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed