BDBM50387537 CHEMBL2057364

SMILES CC(C)(C)NS(=O)(=O)c1cncc(c1)-c1ccc2nc(NC(=O)NCCn3cccn3)nn2c1

InChI Key InChIKey=KFYHKGHTVWFWKP-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50387537   

LigandPNGBDBM50387537(CHEMBL2057364)
Affinity DataIC50: 25.1nMAssay Description:Inhibition of PI3Kgamma in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandPNGBDBM50387537(CHEMBL2057364)
Affinity DataIC50: 200nMAssay Description:Inhibition of PI3Kdelta in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandPNGBDBM50387537(CHEMBL2057364)
Affinity DataIC50: 631nMAssay Description:Inhibition of PI3Kbeta in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandPNGBDBM50387537(CHEMBL2057364)
Affinity DataIC50: 631nMAssay Description:Inhibition of PI3Kalpha in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed