BDBM50389528 CHEMBL2063370

SMILES CCCN(CCC)c1ccc(CC)c2nc(c(C)cc12)-c1c(OC)cc(COC)cc1OC

InChI Key InChIKey=MAPITVFZBHZWOS-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50389528   

LigandPNGBDBM50389528(CHEMBL2063370)
Affinity DataIC50: 115nMAssay Description:Displacement of [125I]-CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandPNGBDBM50389528(CHEMBL2063370)
Affinity DataIC50: 375nMAssay Description:Antagonist activity at human CRF1 receptor expressed in HEK293 cells assessed as inhibition of CRF-stimulated intracellular cAMP accumulation after 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed