BDBM50391028 CHEMBL2088390

SMILES OCc1nc2cc(NC(=O)c3ccc(cc3)C#C)ccc2s1

InChI Key InChIKey=WSWHSSRBYZDUIG-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50391028   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Astrazeneca

Curated by ChEMBL

LigandBDBM50391028(CHEMBL2088390)Copy SMILESCopy InChI

Affinity DataIC50: 175nMAssay Description:Antagonist activity at human recombinant TRPV1 receptor assessed as inhibition of capsaicin-induced calcium uptake by FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
2/8/2013
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL