BDBM50391041 CHEMBL2088407

SMILES Cn1nc(cc1C(=O)Nc1ccc2sc(CO)nc2c1)C(F)(F)F

InChI Key InChIKey=WGOAUHCYBVWDET-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50391041   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Astrazeneca

Curated by ChEMBL

LigandBDBM50391041(CHEMBL2088407)Copy SMILESCopy InChI

Affinity DataIC50: 157nMAssay Description:Antagonist activity at human recombinant TRPV1 receptor assessed as inhibition of capsaicin-induced calcium uptake by FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
2/8/2013
Entry Details Article
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